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SH-I-048A

SH-I-048A (SH-i-048A) is a benzodiazepine derivative related in structure to compounds such as flubromazepam and meclonazepam. SH-I-048A is described as a non subtype selective superagonist at the benzodiazepine site of GABA<sub>A</sub> receptors, with a binding affinity of 0.77&nbsp;nM at the α<sub>1</sub> subtype, 0.17&nbsp;nM at α<sub>2</sub>, 0.38&nbsp;nM at α<sub>3</sub> and 0.11&nbsp;nM at α<sub>5</sub>. It has been used to study the functional differences between the different subtypes of the GABA<sub>A</sub> receptor.

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