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Protein-arginine deiminase

In enzymology, a protein-arginine deiminase (PAD) () is an enzyme that catalyzes a form of post translational modification called arginine de-imination or citrullination:

protein <small>L</small>-arginine + H<sub>2</sub>O protein <small>L</small>-citrulline + NH<sub>3</sub>

Thus, the two substrates of this enzyme are protein <small>L</small>-arginine (arginine residue inside a protein) and H<sub>2</sub>O, whereas its two products are protein <small>L</small>-citrulline and NH<sub>3</sub>:

This enzyme belongs to the family of hydrolases, those acting on carbon-nitrogen bonds other than peptide bonds, specifically in linear amidines. The systematic name of this enzyme class is protein-L-arginine iminohydrolase. This enzyme is also called peptidylarginine deiminase.

Structural studies

As of late 2007, seven structures have been solved for this class of enzymes, with PDB accession codes , , , , , , and .

Mammalian proteins

Mammals have 5 protein-arginine deiminases, with symbols

except for rodents, there the letter case is different:

  • Padi1, Padi2, Padi3, Padi4, Padi6

The different case is just a historical artifact. It doesn't indicate that the rodent proteins are special.

Inhibitors

Irreversible inhibitors

Reversible inhibitors

References