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Noribogainalog

Noribogainalog (nor-IBG), also known as 9-hydroxyibogaminalog, is a drug of the ibogalog family related to noribogaine. It is a simplified analogue of noribogaine.

Pharmacology

The drug acts as a potent serotonin 5-HT<sub>2A</sub> receptor partial agonist ( ≈ 90nM; = 35%). It also has activity as a dopamine transporter (DAT) chaperone. Noribogainalog does not affect locomotor activity, does not produce the head-twitch response, and does not affect various other physiological and behavioral measures. However, it does produce analgesic effects that can be diminished by the serotonin 5-HT<sub>2A</sub> receptor antagonist ketanserin. The drug shows relatively low expected blood–brain barrier permeability.

History

Noribogainalog was first described in the scientific literature by David E. Olson and colleagues by 2021.

See also

References

External links