This is a list of known combined sex-hormonal formulations. Brand names and developmental code names are in parentheses.
Androgens
Injection
Marketed
Veterinary
Marketed
Estrogens
Oral
Marketed
Injection
Marketed
Never marketed
Progestogens
Injection
Marketed
Androgens and estrogens
Oral
Marketed
- Chlorotrianisene/methyltestosterone (Tace mit Androgen)
- Conjugated estrogens/methyltestosterone (Premarin with Methyltestosterone)
- Dienestrol/methyltestosterone (Estan, Lucidon)
- Dienestrol diacetate/methyltestosterone (Farmatest)
- Diethylstilbestrol/methyltestosterone (Tylosterone)
- Esterified estrogens/methyltestosterone (Covaryx, Eemt, Essian, Estratest, Menogen, Syntest)
- Ethinylestradiol/methyltestosterone (Climatone, Dumone, Duotrone, Estandron, Femandren, Femovirin, Gynetone, Lynandron, Mepilin, Mixogen, Primodian)
- Methylestradiol/methyltestosterone (Klimanosid)
- Methylestradiol/methyltestosterone/reserpine (Klimanosid R)
Injection
Marketed
- Estradiol benzoate/testosterone propionate (Bothermon)
- Estradiol benzoate/estradiol dienanthate/testosterone enanthate benzilic acid hydrazone (Climacteron, Lactimex, Lactostat)
- Estradiol benzoate/estradiol phenylpropionate/testosterone propionate/testosterone phenylpropionate/testosterone isocaproate (Estandron Prolongatum, Lynandron Prolongatum, Mixogen [Injection])
- Estradiol benzoate/testosterone isobutyrate (Femandren M, Folivirin)
- Estradiol butyrylacetate/testosterone ketolaurate/reserpine (Klimanosid R-Depot)
- Estradiol cypionate/testosterone cypionate (Depo-Testadiol, Femovirin)
- Estradiol cypionate/testosterone enanthate (Supligol)
- Estradiol valerate/prasterone enanthate (Binodian Depot, Cidodian Depot, Gynodian Depot, Klimax, Supligol NF)
- Estradiol valerate/testosterone enanthate (Deladumone, Despamen, Ditate, Ditate-DS, Gravignost, Primodian Depot, Valertest)
Veterinary
Marketed
Estrogens and progestogens
Oral
Marketed
In birth control pills:
- Drospirenone/estetrol (Nextstellis, Drovelis, Lydisilka)
- Estradiol/nomegestrol acetate (Naemis, Zoely)
- Estradiol valerate/cyproterone acetate (Femilar)
- Estradiol valerate/dienogest (Natazia, Qlaira)
- Ethinylestradiol/chlormadinone acetate (Belara)
- Ethinylestradiol/cyproterone acetate (Diane, Diane-35)
- Ethinylestradiol/desogestrel (Alenvona, Apri, Azurette, Bekyree, Bimizza, Caziant, Cesia, Cimizt, Cyclessa, Cyred, Denise, Desogen, Desirett, Emoquette, Enskyce, Gedarel, Gracial, Isibloom, Juleber, Kalliga, Kariva, Kimidess, Laurina, Linessa, Marvelon, Mercilon, Mircette, Mirvala, Novynette, Ortho-Cept, Pimtrea, Reclipsen, Regulon, Simliya, Solia, Velivet, Viorele, Volnea)
- Ethinylestradiol/dienogest (Valette)
- Ethinylestradiol/dimethisterone (Oracon)
- Ethinylestradiol/drospirenone (Yasmin, Yasminelle, Yaz)
- Ethinylestradiol/drospirenone/levomefolic acid (Beyaz, Safyral)
- Ethinylestradiol/etynodiol diacetate (Demulen)
- Ethinylestradiol/gestodene (Femodene, Femodette, Gynera, Harmonet, Meliane, Minesse, Minulet)
- Ethinylestradiol/levonorgestrel (Amethyst, Aviane, Balcoltra, Falmina, Levlen, Lillow, Orsythia, Vienva)
- Ethinylestradiol/levonorgestrel/bisglycinate
- Ethinylestradiol/levonorgestrel/ferrous fumarate
- Ethinylestradiol/lynestrenol (Lyndiol)
- Ethinylestradiol/medroxyprogesterone acetate (Gianda, Provest)
- Ethinylestradiol/megestrol acetate (Nuvacon, Volidan)
- Ethinylestradiol/norethisterone (Brevicon, Norinyl 1+35, Ortho-Novum 7/7/7, Taytulla, Tri-Norinyl, Zenchent)
- Ethinylestradiol/norethisterone/ferrous fumarate (Blisovi 24 FE, Estrostep Fe, Femcon FE, Kaitlib FE, Lo Minastrin Fe, Loestrin 24 Fe, Microgestin 24 FE)
- Ethinylestradiol/norethisterone acetate (FemHRT)
- Ethinylestradiol/norethisterone acetate/ferrous fumarate
- Ethinylestradiol/norgestimate (Ortho Tri-Cyclen, Sprintec)
- Ethinylestradiol/norgestrel (Ovral)
- Ethinylestradiol/norgestrienone (Miniplanor, Planor)
- Ethinylestradiol/quingestanol acetate (Riglovis)
- Ethinylestradiol sulfonate/norethisterone acetate (Deposiston)
- Mestranol/anagestone acetate (Neo-Novum)
- Mestranol/chlormadinone acetate (C-Quens, Lutedion)
- Mestranol/etynodiol diacetate (Ovulen)
- Mestranol/hydroxyprogesterone acetate (Hormolidin)
- Mestranol/lynestrenol (Lyndiol)
- Mestranol/norethisterone (Norethin, Noriday, Norinyl, Norquen, Ortho-Novum)
- Mestranol/noretynodrel (Enavid, Enovid)
- Quinestrol/etynodiol diacetate (Soluna)
- Quinestrol/levonorgestrel (YuèkÃÂtÃÂng, ÃÂiyuè)
- Quinestrol/norgestrel (Compound Norgestrel)
- Quinestrol/quingestanol acetate (Unovis)
For menopausal hormone therapy and/or gynecological disorders:
- Conjugated estrogens/medrogestone (Presomen)
- Conjugated estrogens/medroxyprogesterone acetate (Prempro, Premphase)
- Conjugated estrogens/norgestrel (Prempak-C)
- Estradiol/drospirenone (Angeliq)
- Estradiol/dydrogesterone (Femoston)
- Estradiol/gestodene (Avaden, Avadene)
- Estradiol/levonorgestrel
- Estradiol/medroxyprogesterone acetate (Indivina, Tridestra)
- Estradiol/norethisterone acetate (Activella, Activelle, Cliane, Estalis, Eviana, Evorel, Kliogest, Novofem)
- Estradiol/norgestimate (Prefest)
- Estradiol/progesterone (Bijuva)
- Estradiol/trimegestone (Lovelle, Totelle)
- Estradiol valerate/cyproterone acetate (Climen, Climen 28)
- Estradiol valerate/estriol/levonorgestrel (CycloÃÂstrogynal)
- Estradiol valerate/levonorgestrel (Cyclo-Progynova N)
- Estradiol valerate/medroxyprogesterone acetate (Dilena, Divina, Divitren, Farludiol, Indivina, Sisare)
- Estradiol valerate/norethisterone (Climagest, Climesse)
- Estradiol valerate/norethisterone acetate (Cliovelle, Norestin, Trisequens)
- Estradiol valerate/norgestrel (Cyclacur, Cyclocur, Cyclo-Progynova, Postoval, Progyluton)
- Ethinylestradiol/ethisterone (Amenorone, Di-Pro, Duosterone, Menstrogen, Oracecron, Orasecron)
- Mestranol/noretynodrel (Enovid)
Never or not yet marketed
In birth control pills:
Transdermal
Marketed
In contraceptive patches:
For menopausal hormone therapy:
Vaginal
Marketed
In contraceptive vaginal rings:
Injection
Marketed
In combined injectable contraceptives:
- Estradiol/megestrol acetate (Mego-E, Chinese Injectable No. 2)
- Estradiol benzoate/estradiol valerate/hydroxyprogesterone caproate (Sin-Ol)
- Estradiol benzoate butyrate/algestone acetophenide (Redimen, Soluna, Unijab)
- Estradiol cypionate/hydroxyprogesterone caproate (Sinbios)
- Estradiol cypionate/medroxyprogesterone acetate (Cyclo-Provera, Cyclofem, Lunelle)
- Estradiol enanthate/algestone acetophenide (Anafertin, Deladroxate, Perlutan, Topasel, Yectames)
- Estradiol valerate/hydroxyprogesterone caproate (Chinese Injectable No. 1)
- Estradiol valerate/norethisterone enanthate (Mesigyna, Mesygest)
For menopausal hormone therapy, gynecological disorders, habitual abortion, and other indications:
Never marketed
In combined injectable contraceptives:
For other indications:
Veterinary
Marketed
Androgens and progestogens
Oral
Marketed
Injection
Marketed
Veterinary
Marketed
Estrogens, progestogens, and androgens
Oral
Marketed
Not yet marketed
Sublingual
Marketed
Injection
Marketed
Never marketed
Veterinary
Marketed
Miscellaneous
Oral
Marketed
Never marketed
Transdermal
Marketed
Vaginal
Marketed
Mixed
Marketed
See also
References