Methylpiperidinopyrazole

Methylpiperidinopyrazole (MPP) is a synthetic, nonsteroidal, and highly selective antagonist of ERα that is used in scientific research to study the function of this receptor. It has 200-fold selectivity for ERα over ERβ and 1000-fold selectivity for blocking ERα-mediated gene transcription relative to that of ERβ.

See also

• Glyceollin
• Propylpyrazoletriol (PPT)
• Diarylpropionitrile (DPN)
• Prinaberel (ERB-041)
• Liquiritigenin
• Menerba
• PHTPP
• (R,R)-Tetrahydrochrysene ((R,R)-THC)

References