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AMG-3

AMG-3 (part of the AM cannabinoid series) is an analgesic drug which is a cannabinoid agonist. It is a derivative of Δ<sup>8</sup>-THC substituted with a dithiolane group on the 3-position side chain. AMG-3 is a potent agonist at both CB<sub>1</sub> and CB<sub>2</sub> receptors with a K<sub>i</sub> of 0.32&nbsp;nM at CB<sub>1</sub> and 0.52&nbsp;nM at CB<sub>2</sub>, and its particularly high binding affinity has led to it being used as a template for further structural development of novel cannabinoid drugs. It has sedative and analgesic effects, with analgesia lasting for up to 36&nbsp;hours after administration.

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